SCHEMBL3266883

SCHEMBL3266883

NC(=O)COC(=O)NC1CCN(c2cccc(-c3ccccc3)n2)CC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 6/20 0.47
SKP1 P63208 6/20 0.47
SKP2 Q13309 6/20 0.47
CNR1 P21554 3/20 0.43
BTK Q06187 1/20 0.41
USP30 Q70CQ3 2/20 0.41
TSHR P16473 1/20 0.40
EPHX1 P07099 1/20 0.40
SMO Q99835 2/20 0.39
HSD11B1 P28845 1/20 0.39
USP2 O75604 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3270072 0.91 SCN9A (0.44) CKS1BSKP1SKP2CNR1BTK
SCHEMBL240063 0.86 CKS1B (0.48) CKS1BSKP1SKP2CNR1
SCHEMBL27629096 0.85 CKS1B (0.53) CKS1BSKP1SKP2CNR1USP30
SCHEMBL3265609 0.84 CKS1B (0.41) CKS1BSKP1SKP2CNR1HSD11B1
SCHEMBL3268988 0.84 HSD11B1 (0.41) CKS1BSKP1SKP2BTKUSP30
SCHEMBL1729064 0.82 CNR1 (0.52) CKS1BSKP1SKP2CNR1USP30
SCHEMBL3266914 0.81 CKS1B (0.49) CKS1BSKP1SKP2BTKUSP30
SCHEMBL3266878 0.77 CKS1B (0.45) CKS1BSKP1SKP2CNR1SMN1; SMN2
SCHEMBL3269143 0.76 CKS1B (0.42) CKS1BSKP1SKP2CNR1TSHR
SCHEMBL3265618 0.76 CNR1 (0.41) CKS1BSKP1SKP2CNR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120004207-A1 THERAPEUTIC USES OF DERIVATIVES OF PIPERIDINYL-AND PIPERIDINYL-ALKYL CARBAMATES SANOFI-AVENTIS (FR) 2012-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120004207-A1 THERAPEUTIC USES OF DERIVATIVES OF PIPERIDINYL-AND PIPERIDINYL-ALKYL CARBAMATES CLCN2, CLIC1, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 CKS1B 1534/4885SKP1 4286/4885SKP2 2651/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.