SCHEMBL3267873

SCHEMBL3267873

CC1=C(C(=O)OCc2ccccc2)C(c2cccs2)c2cn[nH]c2N1.CC1=C(C(=O)OCc2ccccc2)C(c2nccs2)c2cn[nH]c2N1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 1/20 0.50
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
HTT P42858 1/20 0.41
PDE1C Q14123 1/20 0.41
ADORA3 P0DMS8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3000827 0.94 PDE1C (0.45) ADORA2BALDH1A1PDE1CADORA3
SCHEMBL4260613 0.92 ADORA2B (0.57) ADORA2BALDH1A1MEN1MAPTKMT2A
SCHEMBL3004313 0.82 ALDH1A1 (0.56) ADORA2BALDH1A1MEN1MAPTKMT2A
SCHEMBL3002847 0.79 PDE1C (0.54) ALDH1A1KDM4EPDE1CADORA3
SCHEMBL3242915 0.76 PDE1C (0.48) MEN1KMT2APDE1CADORA3
SCHEMBL3241017 0.73 PDE1C (0.59) ALDH1A1MEN1MAPTKMT2AKDM4E
SCHEMBL2996950 0.72 PDE1C (0.45) PDE1CADORA3
SCHEMBL7696472 0.72 ALDH1A1 (0.54) ADORA2BALDH1A1MEN1MAPTKMT2A
SCHEMBL3006899 0.71 PDE1C (0.44) ALDH1A1KDM4EPDE1CADORA3
SCHEMBL3237974 0.69 TSHR (0.44) MAPTPDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010002483-A1 OPTIONALLY CONDENSED DIHYDRO PYRIDINE, DIHYDROPYRIMIDINE AND DIHYDRO PYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2010-01-07 WO disclosed