SCHEMBL3267927

SCHEMBL3267927

Cn1nccc1NC(=O)N1CCN(c2cccc(-c3cccc(F)c3F)n2)CC1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FAAH O00519 7/20 0.50
TRPV1 Q8NER1 4/20 0.43
CSNK1D P48730 1/20 0.41
CSNK1E P49674 1/20 0.41
KDM4E B2RXH2 5/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
MAP4K1 Q92918 1/20 0.38
HSD17B10 Q99714 2/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3269363 0.87 FAAH (0.67) FAAHTRPV1CSNK1DCSNK1EKDM4E
SCHEMBL3268200 0.82 ALDH1A1 (0.56) FAAHTRPV1KDM4EALDH1A1MAPT
SCHEMBL3267735 0.81 CSNK1D (0.47) FAAHCSNK1DCSNK1EMAPTHSD17B10
SCHEMBL3267793 0.80 FAAH (0.53) FAAHTRPV1KDM4EALDH1A1
SCHEMBL3269821 0.80 FAAH (0.76) FAAHTRPV1CSNK1DCSNK1E
SCHEMBL3270509 0.79 FAAH (0.49) FAAHTRPV1KDM4EALDH1A1MAPT
SCHEMBL3270535 0.79 FAAH (0.48) FAAHTRPV1KDM4EALDH1A1MAPT
SCHEMBL3274880 0.79 FAAH (0.57) FAAHTRPV1CSNK1DKDM4EALDH1A1
SCHEMBL3774639 0.78 FAAH (0.67) FAAHALDH1A1MAPTHSD17B10TP53
SCHEMBL13184477 0.76 FAAH (0.43) FAAHTRPV1MAPTMAP4K1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100234389-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-16 US disclosed
US-20100234389-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-16 US disclosed
EP-2199282-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2010-06-23 EP disclosed
US-20090163508-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-25 US disclosed
US-20090163508-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-25 US disclosed
US-20090163508-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100234389-A1 AMIDE COMPOUND FAAH, FAAH2, NAAA FAAH 1/4885TRPV1 6/4885CSNK1D 2982/4885
US-20090163508-A1 AMIDE COMPOUND FAAH, FAAH2, NAAA FAAH 1/4885TRPV1 6/4885CSNK1D 2982/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.