SCHEMBL3269545

SCHEMBL3269545

NC(=O)Oc1[nH]c2ccsc2c1Sc1cccc(Br)c1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TYMS P04818 2/20 0.35
MAPK8 P45983 1/20 0.33
POLB P06746 1/20 0.32
PARP1 P09874 1/20 0.31
KDR P35968 1/20 0.30
ERCC5 P28715 1/20 0.30
FEN1 P39748 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3268577 0.87 KDR (0.39) MAPK8PARP1KDR
SCHEMBL3269989 0.87 KDR (0.39) TYMSMAPK8POLBPARP1KDR
SCHEMBL3268931 0.86 TUBB4A (0.37) POLBKDRMEN1KMT2A
SCHEMBL3275434 0.85 EDNRA (0.43) MAPK8PARP1KDRMEN1KMT2A
SCHEMBL3268815 0.83 TNKS2 (0.38) TYMSMAPK8POLBPARP1MEN1
SCHEMBL3175305 0.83 TYMS (0.37) TYMSMAPK8POLBPARP1KDR
SCHEMBL3269135 0.82 RHEB (0.43) MAPK8FEN1MEN1KMT2A
SCHEMBL3268889 0.81 MAPK8 (0.32) MAPK8PARP1
SCHEMBL3269102 0.81 PDPK1 (0.36) TYMSPOLBPARP1MEN1KMT2A
SCHEMBL3268326 0.79 CCNC (0.33) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784409-B1 SUBSTITUTED THIENOPYRROLE CARBOXYLIC ACID AMIDES, PYRROLOTHIAZOLE CARBOXYLIC ACID AMIDES, AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2010-06-16 EP claimed