SCHEMBL3268326

SCHEMBL3268326

NC(=O)Oc1[nH]c2ccsc2c1Sc1ccncc1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
TYMS P04818 9/20 0.33
DHFR P00374 2/20 0.33
DDAH1 O94760 1/20 0.31
NOS1 P29475 1/20 0.31
CDC7 O00311 1/20 0.31
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP12 P39900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3268931 0.88 TUBB4A (0.37)
SCHEMBL3267982 0.85 MEN1 (0.34) TYMSDHFR
SCHEMBL3269983 0.85 ALDH1A1 (0.34)
SCHEMBL3269102 0.82 PDPK1 (0.36) TYMSDHFR
SCHEMBL3268889 0.82 MAPK8 (0.32)
SCHEMBL3270359 0.81 MMP1 (0.33) MMP1MMP2MMP9MMP12
SCHEMBL3182168 0.81 PTGS2 (0.39) CCNCCDK8TYMSDHFRDDAH1
SCHEMBL3268792 0.81 CDC7 (0.36) CCNCCDK8TYMSDHFRDDAH1
SCHEMBL3268887 0.80 PTGS1 (0.35)
SCHEMBL3269989 0.79 KDR (0.39) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784409-B1 SUBSTITUTED THIENOPYRROLE CARBOXYLIC ACID AMIDES, PYRROLOTHIAZOLE CARBOXYLIC ACID AMIDES, AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2010-06-16 EP claimed