SCHEMBL3270325

SCHEMBL3270325

NC(=O)Oc1[nH]c2ccsc2c1Sc1ccccc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GAA P10253 2/20 0.33
ALDH1A1 P00352 1/20 0.32
SCD O00767 2/20 0.31
PTPN11 Q06124 2/20 0.31
PARP1 P09874 1/20 0.31
CTNNB1 P35222 1/20 0.31
WNT3A P56704 1/20 0.31
HPGD P15428 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3268936 0.87 NPC1 (0.38) HPGD
SCHEMBL3272702 0.86 PDE7A (0.39) KDM4ELMNAMAPTGAAALDH1A1
SCHEMBL3269317 0.85 MEN1 (0.36) HPGD
SCHEMBL3270253 0.83 TUBB4A (0.31) LMNA
SCHEMBL3267800 0.83 TUBB4A (0.42) KDM4EMAPTNPSR1
SCHEMBL3184621 0.82 PARP1 (0.35) KDM4ELMNAMAPTNPSR1GAA
SCHEMBL3268931 0.82 TUBB4A (0.37) NPSR1ALDH1A1HPGD
SCHEMBL3268818 0.81 USP7 (0.36) NPSR1PTPN11
SCHEMBL3270359 0.79 MMP1 (0.33) HPGD
SCHEMBL4038003 0.78 PARP1 (0.39) KDM4ELMNAMAPTNPSR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784409-B1 SUBSTITUTED THIENOPYRROLE CARBOXYLIC ACID AMIDES, PYRROLOTHIAZOLE CARBOXYLIC ACID AMIDES, AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2010-06-16 EP claimed