SCHEMBL3272415

SCHEMBL3272415

NC(=O)Oc1[nH]c2sccc2c1Sc1ccccn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICAM1 P05362 1/20 0.36
SELE P16581 1/20 0.36
VCAM1 P19320 1/20 0.36
TNKS2 Q9H2K2 2/20 0.35
TNKS O95271 1/20 0.35
PARP1 P09874 1/20 0.35
PARP15 Q460N3 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
L3MBTL1 Q9Y468 3/20 0.32
LMNA P02545 2/20 0.32
NPC1 O15118 1/20 0.32
METAP2 P50579 1/20 0.32
RAB9A P51151 1/20 0.32
METAP1 P53582 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KRAS P01116 1/20 0.32
GCK P35557 2/20 0.32
CA2 P00918 1/20 0.31
BRAF P15056 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3167765 0.82 ICAM1 (0.41) ICAM1SELEVCAM1TNKS2TNKS
SCHEMBL3270312 0.82 TNKS2 (0.39) TNKS2TNKSPARP1PARP15PARP2
SCHEMBL3268887 0.82 PTGS1 (0.35) ICAM1SELEVCAM1PTGS1PTGS2
SCHEMBL3835657 0.81 ALDH1A1 (0.43) ICAM1SELEVCAM1PARP1PTGS1
SCHEMBL3268792 0.80 CDC7 (0.36) TNKS2TNKSPARP1PARP15PARP2
SCHEMBL3268877 0.79 PARP15 (0.35) TNKS2TNKSPARP1PARP15ALDH1A1
SCHEMBL4039379 0.78 CHUK (0.42) ICAM1SELEVCAM1PARP1PTGS1
SCHEMBL3274125 0.77 ICAM1 (0.34) ICAM1SELEVCAM1PTGS1PTGS2
SCHEMBL3270015 0.76 TUBB4A (0.42) TNKS2TNKSPARP1PARP15PARP2
SCHEMBL4033284 0.75 PTGS1 (0.37) ICAM1SELEVCAM1PARP1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784409-B1 SUBSTITUTED THIENOPYRROLE CARBOXYLIC ACID AMIDES, PYRROLOTHIAZOLE CARBOXYLIC ACID AMIDES, AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2010-06-16 EP claimed