SCHEMBL4033284

SCHEMBL4033284

NC(=O)Oc1[nH]c2cccnc2c1Sc1ccccn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
PARP1 P09874 5/20 0.36
PDE5A O76074 1/20 0.36
ALDH1A1 P00352 5/20 0.35
PKM P14618 1/20 0.35
DHODH Q02127 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
ICAM1 P05362 1/20 0.34
SELE P16581 1/20 0.34
VCAM1 P19320 1/20 0.34
GCK P35557 1/20 0.33
JAK2 O60674 1/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3835657 0.86 ALDH1A1 (0.43) PTGS1PTGS2PARP1PDE5AALDH1A1
SCHEMBL4035502 0.86 TUBB4A (0.39) PARP1PDE5AALDH1A1DHODHPARP2
SCHEMBL4214923 0.83 ALDH1A1 (0.37) PARP1PDE5AALDH1A1PKMDHODH
SCHEMBL4033192 0.83 PKN1 (0.38) PARP1PDE5APARP2JAK2KCNMA1
SCHEMBL4041978 0.82 CNR2 (0.35) PARP1PDE5AALDH1A1JAK2LMNA
SCHEMBL4036107 0.82 PDE5A (0.36) PARP1PDE5AALDH1A1ICAM1SELE
SCHEMBL4034813 0.82 PKM (0.43) PARP1PDE5AALDH1A1PKMLMNA
SCHEMBL2049930 0.81 PARP1 (0.39) PTGS1PTGS2PARP1ALDH1A1PKM
SCHEMBL4032967 0.81 SMN1; SMN2 (0.41) PDE5AALDH1A1PKMLMNAHPGD
SCHEMBL4039379 0.81 CHUK (0.42) PTGS1PTGS2PARP1ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747220-B1 SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2009-04-15 EP claimed