SCHEMBL327357

SCHEMBL327357

CC(C(=O)OC(C)(C)C)N1CCSCC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PREP P48147 2/20 0.40
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
FDPS P14324 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
USP2 O75604 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HTT P42858 1/20 0.31
ATM Q13315 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
DGAT1 O75907 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6600488 0.79 SIGMAR1 (0.41) HRH3USP2SMN1; SMN2HTTATM
SCHEMBL17025687 0.79 HRH3 (0.35) KMT2AHRH3USP2SMN1; SMN2HTT
SCHEMBL27793003 0.76 ALDH1A1 (0.41) MEN1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL3825201 0.75 HSD17B10 (0.45) MEN1KMT2AHRH3SMN1; SMN2ALDH1A1
SCHEMBL7280643 0.74 PREP (0.33) PREP
SCHEMBL23096731 0.73 HRH3 (0.40) MEN1CYP2D6KMT2AHRH3USP2
SCHEMBL4435334 0.72 FDPS (0.43) MEN1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7419074 0.72 HRH3 (0.37) HRH3KDM4E
SCHEMBL4344525 0.71 HRH3 (0.38) HRH3HTTALDH1A1HPGD
SCHEMBL4337458 0.71 HRH3 (0.38) HRH3HTTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590954-A1 BISARYL (THIO)MORPHOLINE DERIVATIVES AS S1P MODULATORS ABBVIE B.V. (NL) 2013-05-15 EP disclosed
WO-2012004375-A1 BISARYL (THIO)MORPHOLINE DERIVATIVES AS S1P MODULATORS ABBOTT HEALTHCARE PRODUCTS B.V. (NL) 2012-01-12 WO disclosed