SCHEMBL3279652

SCHEMBL3279652

O=C(c1ccccc1)c1c[nH]c2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.79
TP53 P04637 1/20 0.69
SMN1; SMN2 Q16637 1/20 0.69
NPSR1 Q6W5P4 1/20 0.69
CTNNB1 P35222 1/20 0.66
WNT3A P56704 1/20 0.66
ALDH1A1 P00352 2/20 0.62
PBRM1 Q86U86 1/20 0.62
ATM Q13315 1/20 0.62
PIM1 P11309 1/20 0.59
NR4A2 P43354 2/20 0.58
ADAM17 P78536 1/20 0.58
MAPK1 P28482 1/20 0.57
CREBBP Q92793 1/20 0.57
KMT2A Q03164 3/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
MEN1 O00255 2/20 0.55
TDP1 Q9NUW8 1/20 0.55
GABRP O00591 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29988308 1.00 GPR84 (0.79) GPR84TP53SMN1; SMN2NPSR1CTNNB1
SCHEMBL2028344 0.88 GPR84 (1.00) GPR84TP53SMN1; SMN2NPSR1CTNNB1
SCHEMBL6247701 0.88 GPR84 (0.71) GPR84TP53SMN1; SMN2NPSR1CTNNB1
SCHEMBL12707173 0.88 CFTR (0.61) GPR84TP53SMN1; SMN2NPSR1CTNNB1
SCHEMBL22634965 0.87 GPR84 (0.65) GPR84TP53SMN1; SMN2NPSR1CTNNB1
SCHEMBL27694373 0.86 GPR84 (0.69) GPR84TP53SMN1; SMN2NPSR1CTNNB1
SCHEMBL9545117 0.86 GPR84 (0.69) GPR84TP53SMN1; SMN2NPSR1CTNNB1
SCHEMBL6705760 0.86 GPR84 (0.69) GPR84TP53SMN1; SMN2NPSR1CTNNB1
SCHEMBL2980233 0.86 SMN1; SMN2 (0.71) GPR84TP53SMN1; SMN2NPSR1ALDH1A1
SCHEMBL64182 0.84 GPR84 (0.77) GPR84CTNNB1WNT3AALDH1A1PBRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242449-B1 TREATING PROSTATIC HYPERTROPHY, URINATION DISORDERS ASSOCIATED WITH PROSTATIC HYPERTROPHY, MALE PATTERN ALOPECIA, OR ACNE ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-06-05 US claimed
CN-1264365-A 3-benzoylindole derivatives and drugs containing the same ZERIA PHARM CO LTD (JP) 2000-08-23 CN claimed
EP-0997457-A1 3-BENZOYLINDOLE DERIVATIVES AND DRUGS CONTAINING THE SAME ZERIA PHARMACEUTICAL CO., LTD. (JP) 2000-05-03 EP claimed
CN-1049156-A Indenoindole compounds UNIV BATH (GB) 1991-02-13 CN claimed
WO-1990015800-A1 INDENOINDOLE COMPOUNDS UNIVERSITY OF BATH (GB) 1990-12-27 WO claimed
EP-0404536-A1 Indenoindole compounds I UNIVERSITY OF BATH (GB) 1990-12-27 EP claimed
JP-11035558-A None JP disclosed
US-11891386-B2 Indole compounds and their use ARIAGEN, INC. (CA) 2024-02-06 US disclosed
US-20230278986-A1 ARYL HYDROCARBON RECEPTOR MODULATORS AND USES THEREOF BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2023-09-07 US disclosed
US-20230278986-A1 ARYL HYDROCARBON RECEPTOR MODULATORS AND USES THEREOF BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2023-09-07 US disclosed
US-20230278986-A1 ARYL HYDROCARBON RECEPTOR MODULATORS AND USES THEREOF BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2023-09-07 US disclosed
US-20230145074-A1 Indole Compounds and Their Use ARIAGEN, INC. (US) 2023-05-11 US disclosed
US-20230145074-A1 Indole Compounds and Their Use ARIAGEN, INC. (US) 2023-05-11 US disclosed
WO-1999003831-A1 3-BENZOYLINDOLE DERIVATIVES AND DRUGS CONTAINING THE SAME ZERIA PHARMACEUTICAL CO., LTD. (JP) 1999-01-28 WO disclosed
EP-0734386-A1 PLATELET ACTIVATING FACTOR ANTAGONISTS: IMIDAZOPYRIDINE INDOLES Abbott Laboratories (US) 1996-10-02 EP disclosed
US-5486525-A ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES (US) 1996-01-23 US disclosed
WO-1995016687-A1 PLATELET ACTIVATING FACTOR ANTAGONISTS: IMIDAZOPYRIDINE INDOLES ABBOTT LABORATORIES (US) 1995-06-22 WO disclosed
CN-1056685-A Indole derivatives and preparation method thereof FUJISAWA PHARMACEUTICAL CO (JP) 1991-12-04 CN disclosed
US-4731353-A METAL SALT OF INDOLE-2-CARBOXYLIC ACID COLOR DEVELOPER KANZAKI PAPER MANUFACTURING COMPANY, LIMITED (JP) 1988-03-15 US disclosed
US-4110536-A ANTIARRHYTHMIA MILES LABORATORIES, INC. (US) 1978-08-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11891386-B2 Indole compounds and their use IDO1, IDO2, INMT GPR84 801/4885TP53 24/4885SMN1; SMN2 4567/4885
US-20230278986-A1 ARYL HYDROCARBON RECEPTOR MODULATORS AND USES THEREOF AHR, ARNT, NR4A1 GPR84 80/4885TP53 1611/4885SMN1; SMN2 4063/4885
US-20230145074-A1 Indole Compounds and Their Use IDO1, IDO2, INMT GPR84 801/4885TP53 24/4885SMN1; SMN2 4567/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.