Tyrosine

Tyrosine

SCHEMBL3303402

NC(Cc1ccc(O)cc1)C(=O)O.NCCCCC(N)C(=O)O

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Tyrosine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 known ✓ P23219 2/20 0.53
PTGS2 known ✓ P35354 1/20 0.50
SLC7A5 Q01650 3/20 0.73
GSR P00390 1/20 0.61
ITGB3 P05106 1/20 0.59
ITGA2B P08514 1/20 0.59
ALPI P09923 1/20 0.53
PKM P14618 1/20 0.53
XIAP P98170 1/20 0.53
THRB P10828 1/20 0.51
LNPEP Q9UIQ6 2/20 0.50
ERAP2 Q6P179 1/20 0.50
KDM4E B2RXH2 1/20 0.50
USP2 O75604 1/20 0.50
EGFR P00533 1/20 0.50
LCK P06239 1/20 0.50
FYN P06241 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
ALOX15 P16050 1/20 0.50
HTR2A P28223 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tyrosine SCHEMBL3485478 1.00 SLC7A5 (0.73) SLC7A5GSRITGB3ITGA2BPTGS1
Tyrosine SCHEMBL21925058 1.00 SLC7A5 (0.73) SLC7A5GSRITGB3ITGA2BPTGS1
Tyrosine SCHEMBL571284 1.00 SLC7A5 (0.73) SLC7A5GSRITGB3ITGA2BPTGS1
Tyrosine SCHEMBL27709284 0.98 SLC7A5 (0.71) SLC7A5GSRITGB3ITGA2BPTGS1
Tyrosine SCHEMBL22207546 0.96 SLC7A5 (0.67) SLC7A5GSRITGB3ITGA2BPTGS1
Tyrosine SCHEMBL2723438 0.96 SLC7A5 (0.67) SLC7A5GSRITGB3ITGA2BPTGS1
Tyrosine SCHEMBL27074660 0.96 SLC7A5 (0.67) SLC7A5GSRITGB3ITGA2BPTGS1
Tyrosine SCHEMBL22654492 0.96 SLC7A5 (0.67) SLC7A5GSRITGB3ITGA2BPTGS1
Tyrosine SCHEMBL5066575 0.96 SLC7A5 (0.67) SLC7A5GSRITGB3ITGA2BPTGS1
Tyrosine SCHEMBL27765246 0.95 SLC7A5 (0.75) SLC7A5GSRITGB3ITGA2BPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100298227-A1 Treatment of autoimmune conditions with Copolymer 1 and related copolymers President and Fellows of Harvard College and Yeda Research 2010-11-25 US claimed
WO-2002086153-A1 DETERMINING RESISTANCE TO A $G(b)-LACTAM-CONTAINING ANTIBIOTIC BY COMPARING THE RATIO OF TWO $G(b)-LACTAMASE GENES DIATECH PTY LTD (AU) 2002-10-31 WO claimed
CN-109750019-A It is a kind of to improve monocot crops to the method and application of gibberellin inhibitor sensitiveness 中国农业大学 2019-05-14 CN disclosed
US-7741019-B2 Detection of ovarian cancer MOUNT SINAI HOSPITAL (CA) 2010-06-22 US disclosed
CN-1938042-B Use of aromatic cationic peptides for the manufacture of a medicament for the reduction of oxidative damage CORNELL RES FOUNDATION INC 2010-06-02 CN disclosed
US-20090280179-A1 Resorbable Calcium Phosphate Based Biopolymer-Cross-Linked Bone Replacement Material DOT GMBH (DE) 2009-11-12 US disclosed
CN-100536909-C method for preventing mitochondrial permeability transition CORNELL RES FOUNDATION INC CLI (US) 2009-09-09 CN disclosed
CN-101378789-A Reabsorabable calcium phosphate based biopolymer-cross-linked bone replacement material DOT GMBH (DE) 2009-03-04 CN disclosed
CN-101214380-A Method and carrier complexes for delivering molecules to cells CORNELL RES FOUNDATION INC (US) 2008-07-09 CN disclosed
US-7204997-B2 Responsive microgel and methods related thereto SUPRATEK PHARMA INC. (CA) 2007-04-17 US disclosed
US-20060223059-A1 Methods for detecting endocrine cancer MOUNT SINAI HOSPITAL (CA) 2006-10-05 US disclosed
EP-1330652-A2 METHOD FOR DETECTING OVARIAN CANCER BASED ON HUMAN KALLIKREIN 6 (HK6) MOUNT SINAI HOSPITAL (CA) 2003-07-30 EP disclosed
WO-2003034068-A1 LOCALIZATION OF DISORDERS ASSOCIATED WITH KALLIKREINS MOUNT SINAI HOSPITAL (CA) 2003-04-24 WO disclosed
WO-2003033731-A2 METHODS FOR DETECTING OVARIAN CANCER MOUNT SINAI HOSPITAL (CA) 2003-04-24 WO disclosed
WO-2002097438-A1 METHOD OF DETECTING AND MONITORING PROSTATE AND OVARIAN CANCERS MOUNT SINAI HOSPITAL (CA) 2002-12-05 WO disclosed
WO-2002086153-A1 DETERMINING RESISTANCE TO A $G(b)-LACTAM-CONTAINING ANTIBIOTIC BY COMPARING THE RATIO OF TWO $G(b)-LACTAMASE GENES DIATECH PTY LTD (AU) 2002-10-31 WO disclosed
WO-2002037112-A2 DETECTION OF OVARIAN CANCER MOUNT SINAI HOSPITAL (CA) 2002-05-10 WO disclosed
WO-2002035232-A2 METHOD FOR DETECTING OVARIAN CANCER BASED ON HUMAN KALLIKREIN 6 (HK6) MOUNT SINAI HOSPITAL (CA) 2002-05-02 WO disclosed
US-5141870-A Transforming plants with mutant fragment confers herbicide resistance E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-08-25 US disclosed
US-4153687-A Derivatives, having an inhibitory action against protease and an antiphlogistic action, of the trypsin-kallikrein inhibitor obtained from cattle organs (BPTI), their preparation and their use as medicaments BAYER AKTIENGESELLSCHAFT (DE) 1979-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090280179-A1 Resorbable Calcium Phosphate Based Biopolymer-Cross-Linked Bone Replacement Material BMP2, BMP4, PLOD3 PTGS1 2624/4885PTGS2 3176/4885SLC7A5 2072/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.