SCHEMBL3306752

SCHEMBL3306752

Nc1nc(Oc2ccc(Br)cc2)c2[nH]cnc2n1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 4/20 0.67
MGMT P16455 8/20 0.56
CDK1 P06493 13/20 0.55
CCNB1 P14635 13/20 0.55
CCNA2 P20248 12/20 0.55
CDK2 P24941 12/20 0.55
CCNA1 P78396 12/20 0.55
LMNA P02545 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 1/20 0.52
NFKB1 P19838 1/20 0.52
CYP2C19 P33261 1/20 0.52
BLM P54132 1/20 0.52
PMP22 Q01453 1/20 0.52
PDPK1 O15530 1/20 0.49
GDA Q9Y2T3 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29460225 0.85 CDK1 (0.66) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL9682546 0.85 CDK1 (0.66) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL3302326 0.81 PIN1 (1.00) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL8619367 0.75 CDK1 (0.66) PIN1MGMTCDK1CCNB1CCNA2
Methylguanine SCHEMBL29903462 0.73 CDK1 (0.69) PIN1MGMTCDK1CCNB1CCNA2
Methylguanine SCHEMBL231097 0.73 CDK1 (0.69) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL16145749 0.71 BRAF (0.72) PIN1
SCHEMBL355362 0.71 PDPK1 (0.66) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL5201806 0.71 CDK1 (0.65) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL8618498 0.71 CDK1 (0.77) PIN1MGMTCDK1CCNB1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8791081-B2 MGMT inhibitor combination for the treatment of neoplastic disorders CASE WESTERN RESERVE UNIVERSITY (US) 2014-07-29 US disclosed
US-20100093647-A1 MGMT INHIBITOR COMBINATION FOR THE TREATMENT OF NEOPLASTIC DISORDERS LIU LILI 2010-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093647-A1 MGMT INHIBITOR COMBINATION FOR THE TREATMENT OF NEOPLASTIC DISORDERS MGMT, MSH2, UNG PIN1 2059/4885MGMT 1/4885CDK1 566/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.