SCHEMBL9682546

SCHEMBL9682546

Nc1nc(Oc2ccccc2)c2[nH]cnc2n1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 12/20 0.66
CCNB1 P14635 12/20 0.66
CCNA2 P20248 12/20 0.66
CDK2 P24941 12/20 0.66
CCNA1 P78396 12/20 0.66
MGMT P16455 7/20 0.66
PIN1 Q13526 7/20 0.66
LMNA P02545 1/20 0.66
CYP1A2 P05177 1/20 0.66
CYP3A4 P08684 1/20 0.66
CYP2D6 P10635 1/20 0.66
CYP2C9 P11712 1/20 0.66
TSHR P16473 1/20 0.66
NFKB1 P19838 1/20 0.66
CYP2C19 P33261 1/20 0.66
BLM P54132 1/20 0.66
PMP22 Q01453 1/20 0.66
PDPK1 O15530 1/20 0.51
GDA Q9Y2T3 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29460225 1.00 CDK1 (0.66) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL3306752 0.85 PIN1 (0.67) CDK1CCNB1CCNA2CDK2CCNA1
6-O-Benzylguanine SCHEMBL31517079 0.79 PIN1 (1.00) CDK1CCNB1CCNA2CDK2CCNA1
6-O-Benzylguanine SCHEMBL61740 0.79 PIN1 (1.00) CDK1CCNB1CCNA2CDK2CCNA1
6-O-Benzylguanine SCHEMBL4631744 0.78 PIN1 (0.97) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8619367 0.77 CDK1 (0.66) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL851965 0.76 PIN1 (0.78) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL2930276 0.76 CDK1 (0.62) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL9458749 0.76 ADORA3 (0.55) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL9681378 0.76 TRPA1 (0.43) CDK1CCNB1CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5153318-A Viricides for hepatitis and human t-cell leukemia/lymphoma viruses BURROUGHS WELLCOME CO. (US) 1992-10-06 US disclosed
EP-0421739-A1 3'-azido purine nucleoside THE WELLCOME FOUNDATION LIMITED (GB) 1991-04-10 EP disclosed