SCHEMBL3311920

SCHEMBL3311920

CCOC(=O)C1CCC(=O)N1Cc1cc(OC)c(C(C)(C)C)cc1-c1cccnc1OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GYS1 P13807 1/20 0.39
POLB P06746 1/20 0.37
HCRTR1 O43613 3/20 0.36
HCRTR2 O43614 3/20 0.36
AGTR2 P50052 1/20 0.36
ADRA1A P35348 2/20 0.35
MAPT P10636 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1B P35368 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3311912 1.00 GYS1 (0.39) GYS1POLBHCRTR1HCRTR2AGTR2
SCHEMBL2347999 0.86 HCRTR1 (0.38) GYS1HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL2347996 0.86 HCRTR1 (0.38) GYS1HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL3315063 0.82 HCRTR1 (0.36) GYS1HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL3315057 0.81 HCRTR1 (0.36) GYS1HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL3315053 0.80 HCRTR1 (0.35) GYS1HCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL2364233 0.80 ADRA1A (0.37) GYS1POLBHCRTR1HCRTR2ADRA1A
SCHEMBL2364234 0.80 ADRA1A (0.37) GYS1POLBHCRTR1HCRTR2ADRA1A
SCHEMBL11949287 0.79 ALOX5AP (0.38) KDM4EALDH1A1
SCHEMBL11949290 0.78 PDE4B (0.37) HCRTR1HCRTR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8232271-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2012-07-31 US disclosed
US-20100111900-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS ROCHE PALO ALTO LLC 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100111900-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS POLR2A, EIF2AK2, POLR2B GYS1 3878/4885POLB 16/4885HCRTR1 1471/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.