SCHEMBL3344813

SCHEMBL3344813

CC(Cc1ccccn1)c1cc(C#N)c(N)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
MAPT P10636 5/20 0.37
HPGD P15428 2/20 0.37
TSHR P16473 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TP53 P04637 1/20 0.37
ALOX15 P16050 1/20 0.37
HBB P68871 1/20 0.37
SLC22A12 Q96S37 4/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
MCL1 Q07820 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3349055 0.75 CHRM2 (0.40) MAPTHPGDTSHRSMN1; SMN2RAB9A
SCHEMBL3344814 0.75 MEN1 (0.34) ADORA2AADORA1MAPTHPGDTSHR
SCHEMBL3299360 0.75 L3MBTL1 (0.42) ADORA2AADORA1MAPTHPGDTSHR
SCHEMBL3304121 0.70 ADORA2A (0.46) ADORA2AADORA1MAPTHPGDSMN1; SMN2
SCHEMBL4847045 0.70 GRM6 (0.32) MAPTHPGDTSHRSMN1; SMN2ALDH1A1
SCHEMBL3301341 0.69 ALDH1A1 (0.39) ADORA2AADORA1MAPTHPGDSMN1; SMN2
SCHEMBL2369914 0.67 GRIN2D (0.47) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL11338065 0.66 GRIN2D (0.47) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL10087892 0.65 GRIN2D (0.62) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL24454696 0.65 GRIN2D (0.61) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045015-A1 HETEROARYL SUBSTITUTED THIENO[2,3-D]PYRIMIDINE AND THEIR USE AS ADENOSINE A2A RECEPTOR ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2010-04-22 WO disclosed