SCHEMBL3345101

SCHEMBL3345101

Cc1cc(-c2nc(N)c3cc(C(=O)O)sc3n2)no1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 1/20 0.43
ADORA2A P29274 13/20 0.41
ADORA1 P30542 10/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 1/20 0.39
MEN1 O00255 1/20 0.37
GLA P06280 1/20 0.37
PKM P14618 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
POLB P06746 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PDE8B O95263 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3302932 0.82 RAB9A (0.46) ADORA2AADORA1KDM4EALDH1A1GAA
SCHEMBL3302092 0.76 TSHR (0.55) ADORA2AADORA1KDM4EALDH1A1MEN1
SCHEMBL3302089 0.75 CHRM4 (0.46) ADORA2AADORA1GAAMEN1KMT2A
SCHEMBL3348239 0.74 ADORA2A (0.70) HSP90AB1ADORA2AADORA1KDM4EALDH1A1
SCHEMBL3351882 0.72 ADORA2A (0.59) HSP90AB1ADORA2AADORA1
SCHEMBL3303592 0.68 ADORA2A (0.66) ADORA2AADORA1
SCHEMBL31044888 0.66 KDM4E (0.33) ADORA2AADORA1KDM4EALDH1A1GAA
SCHEMBL3351568 0.66 ADORA2A (0.75) ADORA2AADORA1
SCHEMBL13780035 0.64 KDM4E (0.51) HSP90AB1KDM4EALDH1A1MEN1GLA
SCHEMBL5456062 0.64 HSP90AB1 (0.45) HSP90AB1KDM4EALDH1A1GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045008-A1 AMIDES OF THIENO[2,3-d]PYRIMIDINE AND THEIR USE AS ADENOSINE A2a RECEPTOR ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2010-04-22 WO disclosed