SCHEMBL3345200

SCHEMBL3345200

COCCOc1cc(N2CCN(CC=O)CC2)ccc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.41
RAD52 P43351 1/20 0.41
HTR1A P08908 5/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM1A O60341 1/20 0.37
ADORA2B P29275 3/20 0.35
HTR4 Q13639 3/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
RECQL P46063 1/20 0.35
PTK2B Q14289 1/20 0.35
ADORA2A P29274 3/20 0.35
ADORA1 P30542 1/20 0.35
KCNH2 Q12809 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2726089 0.86 ALDH1A1 (0.48) GAARAD52ALDH1A1ADORA2BHTR4
SCHEMBL3346276 0.82 MAPT (0.55) ALDH1A1KDM4EMAPTMAPK1HTT
SCHEMBL3349822 0.81 GAA (0.43) GAARAD52ALDH1A1KDM4EMAPT
SCHEMBL3309942 0.80 CASP6 (0.51) ALDH1A1MAPT
SCHEMBL3345906 0.79 GAA (0.44) GAARAD52ALDH1A1KDM4EMAPT
SCHEMBL16935878 0.75 MAP4K4 (0.44) HTR1ADRD3
SCHEMBL17265652 0.75 GAA (0.49) GAARAD52ALDH1A1KDM4EMAPT
SCHEMBL310404 0.75 HTR4 (0.48) GAARAD52HTR1AADORA2BHTR4
SCHEMBL15994391 0.74 MAPT (0.46) GAARAD52HTR1AALDH1A1ADORA2B
SCHEMBL17265647 0.74 CYP1A2 (0.51) GAARAD52ALDH1A1HTR4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010049731-A1 PYRAZOLO- AND IMIDAZOPYRIDINYLPYRIMIDINEAMINES AS IGF-1R TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-05-06 WO disclosed