SCHEMBL3345216

SCHEMBL3345216

COc1cc(N2CCN(CC=O)CC2)c(OC)cc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
MAPT P10636 2/20 0.47
ALDH1A3 P47895 1/20 0.40
HTR4 Q13639 4/20 0.39
ADORA2B P29275 3/20 0.39
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
DRD4 P21917 1/20 0.38
DRD2 P14416 1/20 0.37
KDM4E B2RXH2 2/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
DRD1 P21728 1/20 0.36
DRD3 P35462 1/20 0.36
GLA P06280 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346862 0.89 ALDH1A1 (0.39) ALDH1A1MAPTALDH1A3HTR4ADORA2B
SCHEMBL3344767 0.88 ALDH1A1 (0.39) ALDH1A1MAPTHTR4ADORA2BKDM4E
SCHEMBL20591936 0.82 ALDH1A1 (0.48) ALDH1A1MAPTALDH1A3ADRA1DADRA1A
SCHEMBL2726089 0.80 ALDH1A1 (0.48) ALDH1A1MAPTHTR4ADORA2BKDM4E
SCHEMBL3345838 0.79 ALDH1A1 (0.48) ALDH1A1MAPTKDM4ELMNAHTT
SCHEMBL1911914 0.77 DRD2 (0.53) ALDH1A1MAPTDRD2KDM4EHTT
SCHEMBL20764155 0.77 MAPT (0.58) ALDH1A1MAPTALDH1A3KDM4ELMNA
SCHEMBL10810169 0.76 ALDH1A1 (0.57) ALDH1A1MAPTALDH1A3KDM4ELMNA
SCHEMBL1193917 0.75 DRD2 (0.64) ALDH1A1MAPTADRA1DADRA1AADRA1B
SCHEMBL3346311 0.75 KDM4E (0.36) ALDH1A1MAPTALDH1A3ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010049731-A1 PYRAZOLO- AND IMIDAZOPYRIDINYLPYRIMIDINEAMINES AS IGF-1R TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-05-06 WO disclosed