SCHEMBL3345353

SCHEMBL3345353

Cn1c(=O)ccc2ncc(F)c(OC[C@H]3CC[C@H](NC(=O)O)CC3)c21

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 8/20 0.41
HPGD P15428 1/20 0.35
HRH3 Q9Y5N1 2/20 0.35
DHODH Q02127 1/20 0.35
RORC P51449 1/20 0.35
KCNH2 Q12809 1/20 0.34
GRIN2B Q13224 2/20 0.34
SSTR4 P31391 1/20 0.34
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
MAPK8 P45983 1/20 0.34
MAPK9 P45984 1/20 0.34
MAPK10 P53779 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3345358 1.00 LRRK2 (0.41) LRRK2HPGDHRH3DHODHRORC
SCHEMBL3345752 0.92 LRRK2 (0.39) LRRK2HRH3RORCGRIN2BCYP4F2
SCHEMBL3345749 0.92 LRRK2 (0.39) LRRK2HRH3RORCGRIN2BCYP4F2
SCHEMBL3347085 0.88 RORC (0.40) HRH3RORCKCNH2
SCHEMBL3347090 0.88 RORC (0.40) HRH3RORCKCNH2
SCHEMBL3352394 0.87 KCNH2 (0.41) LRRK2RORCKCNH2SSTR4
SCHEMBL3352400 0.87 KCNH2 (0.41) LRRK2RORCKCNH2SSTR4
SCHEMBL3352185 0.85 LRRK2 (0.39) LRRK2HPGDSSTR4MAPK8MAPK9
SCHEMBL3352192 0.85 LRRK2 (0.39) LRRK2HPGDSSTR4MAPK8MAPK9
SCHEMBL3375050 0.83 TLR9 (0.40) LRRK2HRH3RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046388-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUINOLIN-2-ONES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed
WO-2010045987-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUIN0LIN-2-0NES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed