SCHEMBL3345855

SCHEMBL3345855

Cc1cc2nc(CCC#Cc3sccc3C)ccn2n1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
HTT P42858 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP2A6 P11509 1/20 0.32
FFAR1 O14842 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347052 0.83 CYP2A6 (0.37) ALDH1A1CYP2A6FFAR1
SCHEMBL3347231 0.82 GRM5 (0.35) KDM4EHTTALDH1A1MAPK1L3MBTL1
SCHEMBL3345927 0.80 GRM5 (0.36) CYP1A2CYP2D6
SCHEMBL3347664 0.80 GRM5 (0.37) KDM4EHTTALDH1A1MAPK1L3MBTL1
SCHEMBL3351706 0.79 KDM4E (0.34) KDM4EHTTALDH1A1MAPK1L3MBTL1
SCHEMBL3345928 0.79 GRM5 (0.36) KDM4EHTTALDH1A1MAPK1L3MBTL1
SCHEMBL3346740 0.79 KDM4E (0.32) KDM4EHTTALDH1A1MAPK1L3MBTL1
SCHEMBL3347660 0.78 KDM4E (0.31) KDM4EHTTALDH1A1MAPK1L3MBTL1
SCHEMBL3347285 0.77 KDM4E (0.37) KDM4EHTTALDH1A1MAPK1L3MBTL1
SCHEMBL3351704 0.77 KDM4E (0.34) KDM4EHTTALDH1A1MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed