SCHEMBL3345928

SCHEMBL3345928

Cc1cc2nc(CCC#Cc3ccccc3)ccn2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 9/20 0.36
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HRH3 Q9Y5N1 1/20 0.33
PDE10A Q9Y233 4/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
THPO P40225 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
TP53 P04637 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347641 0.89 GRM5 (0.38) GRM5ALDH1A1KDM4EMAPK1HTT
SCHEMBL3346940 0.87 GRM5 (0.42) GRM5ALDH1A1KDM4EMAPK1HTT
SCHEMBL3345594 0.87 GRM5 (0.40) GRM5ALDH1A1KDM4EMAPK1HTT
SCHEMBL3347306 0.87 CHRNB2 (0.44) GRM5CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3351706 0.85 KDM4E (0.34) GRM5ALDH1A1KDM4EMAPK1HTT
SCHEMBL3347055 0.83 GRM5 (0.51) GRM5ALDH1A1KDM4EMAPK1HTT
SCHEMBL3346926 0.83 GRM5 (0.38) GRM5ALDH1A1KDM4EMAPK1HTT
SCHEMBL3347664 0.83 GRM5 (0.37) GRM5ALDH1A1KDM4EMAPK1HTT
SCHEMBL3347585 0.83 GRM5 (0.34) GRM5ALDH1A1KDM4EMAPK1HTT
SCHEMBL3346856 0.83 GRM5 (0.52) GRM5ALDH1A1KDM4EMAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed