SCHEMBL3346412

SCHEMBL3346412

O=C(NCCc1ccccc1F)[C@@H]1CNC[C@H]1c1ccc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.53
MC4R P32245 3/20 0.45
KCNH2 Q12809 3/20 0.43
REN P00797 1/20 0.43
CYP3A4 P08684 1/20 0.43
ROCK2 O75116 3/20 0.42
CDC42 P60953 1/20 0.42
PRKCE Q02156 1/20 0.42
PRKG2 Q13237 1/20 0.42
PKN2 Q16513 1/20 0.42
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22179085 0.84 MC4R (0.58) CNR1MC4RKDM4EHSD17B10
SCHEMBL3346376 0.84 MC4R (0.63) CNR1MC4RKCNH2HSD17B10
Hydrochloric Acid SCHEMBL22160560 0.83 MC4R (0.57) CNR1MC4RKDM4EHSD17B10
SCHEMBL3347924 0.82 TAAR1 (0.52) CNR1MC4RKCNH2ROCK2HSD17B10
SCHEMBL3380087 0.81 MC4R (0.66) MC4R
SCHEMBL3345900 0.81 KCNH2 (0.58) MC4RKCNH2KDM4EHSD17B10
SCHEMBL3353041 0.81 CNR1 (0.55) CNR1MC4RKCNH2ROCK2CDC42
SCHEMBL3348201 0.79 CNR1 (0.54) CNR1MC4RROCK2KDM4E
Hydrochloric Acid SCHEMBL28625482 0.78 MC4R (0.51) CNR1MC4RKDM4EHSD17B10
SCHEMBL3350700 0.76 ROCK2 (0.42) MC4RKCNH2ROCK2CDC42PRKCE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed