SCHEMBL3346663

SCHEMBL3346663

Cc1cccc(CCNC(=O)[C@@H]2CNC[C@H]2c2ccc(Cl)nc2)n1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.41
KMT2A Q03164 2/20 0.38
ROCK2 O75116 4/20 0.37
MC4R P32245 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.35
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347825 0.88 GPBAR1 (0.43) KCNH2ROCK2MC4RGPBAR1
SCHEMBL3410485 0.83 MC4R (0.43) KCNH2ROCK2MC4RALDH1A1
SCHEMBL3346548 0.83 GPBAR1 (0.39) KMT2AROCK2MC4RKDM4EMEN1
SCHEMBL3410126 0.82 MC4R (0.57) KCNH2MC4RCHRNB2CHRNB4CHRNA3
SCHEMBL3348171 0.80 TAAR1 (0.53) KCNH2KMT2AMC4RKDM4EMEN1
SCHEMBL3353112 0.79 MC4R (0.43) KCNH2ROCK2MC4RCHRNB2CHRNB4
SCHEMBL3346658 0.79 KCNH2 (0.40) KCNH2KMT2AROCK2CHRNB2CHRNB4
SCHEMBL3352433 0.79 CNR1 (0.46) KCNH2KMT2AROCK2MC4RMEN1
SCHEMBL3353146 0.78 TAAR1 (0.47) KCNH2KMT2AROCK2MC4RMEN1
SCHEMBL3346268 0.75 KCNH2 (0.55) KCNH2MC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed