SCHEMBL3352433

SCHEMBL3352433

COc1cccc(CCNC(=O)[C@@H]2CNC[C@H]2c2ccc(Cl)nc2)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.46
ROCK2 O75116 2/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
ROCK1 Q13464 1/20 0.43
GPR39 O43194 1/20 0.42
MC4R P32245 2/20 0.42
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
KCNH2 Q12809 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3410485 0.88 MC4R (0.43) CNR1ROCK2MC4RKCNH2RAB9A
SCHEMBL3348171 0.88 TAAR1 (0.53) CNR1MEN1KMT2AMC4RKCNH2
SCHEMBL3346278 0.88 CNR1 (0.57) CNR1ROCK2CA1CA2MC4R
SCHEMBL3353235 0.86 ROCK2 (0.49) CNR1ROCK2CA1CA2GPR39
SCHEMBL3353112 0.86 MC4R (0.43) CNR1ROCK2MC4RKCNH2RAB9A
SCHEMBL3347960 0.86 CNR1 (0.52) CNR1ROCK2MEN1KMT2ACA1
SCHEMBL3410126 0.85 MC4R (0.57) MC4RKCNH2RAB9A
SCHEMBL3348187 0.84 KCNH2 (0.48) CNR1CA1CA2MC4RMTNR1A
SCHEMBL3346695 0.84 CNR1 (0.50) CNR1ROCK2CA1CA2ROCK1
SCHEMBL3346496 0.81 KCNH2 (0.56) CNR1MEN1KMT2ACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed