SCHEMBL3346548

SCHEMBL3346548

Cc1cccc(CCNC(=O)[C@@H]2CNC[C@H]2c2ccc(Cl)cn2)n1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.39
TRPM5 Q9NZQ8 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MC4R P32245 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 3/20 0.36
ROCK2 O75116 1/20 0.35
FPR3 P25089 1/20 0.35
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
TAAR1 Q96RJ0 2/20 0.34
CASP1 P29466 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GLA P06280 1/20 0.33
JAK1 P23458 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3350852 0.88 MC4R (0.37) TRPM5MC4RROCK2FPR3
SCHEMBL3347825 0.86 GPBAR1 (0.43) GPBAR1MC4RROCK2
SCHEMBL3346450 0.85 FPR3 (0.48) RAB9AMC4RKDM4EALDH1A1ROCK2
SCHEMBL3346663 0.83 KCNH2 (0.41) GPBAR1MC4RKDM4EMEN1KMT2A
SCHEMBL3349714 0.82 MC4R (0.57) NPC1RAB9AMC4RALDH1A1LMNA
SCHEMBL3350808 0.81 TAAR1 (0.53) NPC1RAB9AMC4RKDM4EMEN1
SCHEMBL3346544 0.79 TRPM5 (0.38) TRPM5ROCK2MAPK1
SCHEMBL3346695 0.79 CNR1 (0.50) MC4RALDH1A1ROCK2TAAR1GLA
SCHEMBL3350885 0.78 TAAR1 (0.47) GPBAR1NPC1RAB9AMC4RKDM4E
SCHEMBL21036525 0.72 PTK2 (0.36) TRPM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed