SCHEMBL3346876

SCHEMBL3346876

N#Cc1cccc(CC#Cc2ccn3nccc3n2)c1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
HRH3 Q9Y5N1 1/20 0.37
IDH1 O75874 1/20 0.36
NOS1 P29475 2/20 0.36
ALDH1A1 P00352 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347261 0.83 GRM5 (0.47)
SCHEMBL3348379 0.82 CYP11B1 (0.38) CYP11B1CYP11B2IDH1NOS1ALDH1A1
SCHEMBL3346817 0.82 DYRK1A (0.41) CYP19A1CYP11B1CYP11B2
SCHEMBL3345883 0.82 DYRK1A (0.37) CYP19A1
SCHEMBL3345949 0.80 GRM5 (0.42) IDH1ALDH1A1
SCHEMBL3345830 0.78 FFAR1 (0.40) CYP11B1CYP11B2
SCHEMBL3346993 0.75 GRM5 (0.51)
SCHEMBL2177472 0.73 DYRK1A (0.44) ALDH1A1
SCHEMBL3347519 0.71 GRM4 (0.46) ALDH1A1
SCHEMBL3346985 0.71 GRM5 (0.42) IDH1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO claimed
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed