SCHEMBL3346918

SCHEMBL3346918

C#Cc1ccsc1-c1ccn2nccc2n1.Cc1cc2cc-2c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.41
SCN5A Q14524 1/20 0.36
TGFBR1 P36897 2/20 0.35
ALDH1A1 P00352 3/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
PIK3CD O00329 1/20 0.33
CYP2C9 P11712 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.32
MAPT P10636 2/20 0.31
POLB P06746 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
S100A4 P26447 1/20 0.30
RAD52 P43351 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347243 0.90 DYRK1A (0.44) DYRK1ASCN5ATGFBR1ALDH1A1HPGD
SCHEMBL3346218 0.88 DYRK1A (0.42) DYRK1ASCN5ATGFBR1ALDH1A1HPGD
SCHEMBL3346989 0.86 DYRK1A (0.39) DYRK1ASCN5ATGFBR1ALDH1A1HPGD
SCHEMBL3346482 0.85 DYRK1A (0.45) DYRK1ASCN5ATGFBR1ALDH1A1HPGD
SCHEMBL3347294 0.84 DYRK1A (0.42) DYRK1ASCN5ATGFBR1ALDH1A1HPGD
SCHEMBL3351413 0.83 DYRK1A (0.40) DYRK1ASCN5ATGFBR1ALDH1A1HPGD
SCHEMBL3346924 0.77 PDE2A (0.32) S100A4RAD52
SCHEMBL5946566 0.73 DYRK1A (0.67) DYRK1ASCN5ATGFBR1ALDH1A1KDM4E
SCHEMBL3348367 0.66 CDK2 (0.33)
SCHEMBL3351756 0.64 CCNE1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed