SCHEMBL3350804

SCHEMBL3350804

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(Cl)cn1)c1cccc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 11/20 0.41
KCNH2 Q12809 1/20 0.39
KIT P10721 3/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
NTSR1 P30989 1/20 0.38
WDR5 P61964 2/20 0.37
S1PR2 O95136 1/20 0.37
S1PR3 Q99500 1/20 0.37
MAPK3 P27361 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13365057 0.92 KCNH2 (0.38) MAPK1KCNH2KITROCK2S1PR2
SCHEMBL3380842 0.91 KCNH2 (0.40) MAPK1KCNH2KITROCK2ROCK1
SCHEMBL3349710 0.91 KCNQ3 (0.46) KCNH2NTSR1
SCHEMBL3346689 0.90 POLB (0.50) KITROCK2ROCK1
SCHEMBL3346383 0.89 KCNH2 (0.50) MAPK1KCNH2KITROCK2ROCK1
SCHEMBL3350882 0.85 KCNH2 (0.46) MAPK1KCNH2KIT
SCHEMBL3348168 0.83 KCNH2 (0.45) MAPK1KCNH2KITROCK2MAPK3
SCHEMBL3346544 0.82 TRPM5 (0.38) MAPK1KCNH2ROCK2
SCHEMBL3346446 0.82 ROCK2 (0.42) MAPK1KCNH2ROCK2S1PR3
SCHEMBL13365050 0.81 SSTR4 (0.39) MAPK1KCNH2ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed