SCHEMBL3348921

SCHEMBL3348921

O=C(O)c1cn2nccc2nc1-c1ccc(C#Cc2cccc(F)c2)s1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.39
PTPRC P08575 1/20 0.36
PTPN2 P17706 1/20 0.36
PTPN1 P18031 1/20 0.36
PTPN6 P29350 1/20 0.36
PTPN9 P43378 1/20 0.36
DUSP3 P51452 1/20 0.36
PTPN11 Q06124 1/20 0.36
PTPN22 Q9Y2R2 1/20 0.36
GRM5 P41594 15/20 0.35
HAO1 Q9UJM8 2/20 0.34
DHODH Q02127 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346431 0.89 PTPRC (0.36) PTPRCPTPN2PTPN1PTPN6PTPN9
SCHEMBL3354223 0.80 GRM5 (0.40) GRM5HAO1
SCHEMBL3354005 0.79
SCHEMBL3347271 0.77 DYRK1A (0.42) IKBKBGRM5
SCHEMBL3351328 0.77 CYP2A6 (0.34)
SCHEMBL3345910 0.67 GRM5 (0.35) IKBKBGRM5
SCHEMBL25331092 0.66 ALDH1A1 (0.44) DHODH
SCHEMBL9903113 0.66 KIT (0.44) GRM5
SCHEMBL3347239 0.65 DYRK1A (0.45) GRM5
SCHEMBL5263475 0.65 SALL4 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed