SCHEMBL3351328

SCHEMBL3351328

Cc1ccsc1C#Cc1ccc(-c2nc3ccnn3cc2C(=O)O)s1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.34
FFAR1 O14842 1/20 0.33
PIM1 P11309 1/20 0.30
PIM3 Q86V86 1/20 0.30
PLK3 Q9H4B4 1/20 0.30
PIM2 Q9P1W9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3354223 0.82 GRM5 (0.40) FFAR1
SCHEMBL3354005 0.77
SCHEMBL3347616 0.77 DYRK1A (0.40) CYP2A6
SCHEMBL3348921 0.77 IKBKB (0.39)
SCHEMBL3346431 0.77 PTPRC (0.36)
SCHEMBL25331092 0.66 ALDH1A1 (0.44)
SCHEMBL3346563 0.66 CYP2A6 (0.45) CYP2A6FFAR1
SCHEMBL3353912 0.65 ALDH1A1 (0.31)
SCHEMBL3347604 0.65 PIM1 (0.30) PIM1PIM3PLK3PIM2
SCHEMBL3347071 0.65 CYP2A6 (0.32) CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed