SCHEMBL3348980

SCHEMBL3348980

C[Si](C)(C)C#Cc1cncc(-c2cccnc2)c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.56
CYP2A6 P11509 3/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP11B2 P19099 5/20 0.44
MKNK1 Q9BUB5 2/20 0.41
MKNK2 Q9HBH9 2/20 0.41
MEN1 O00255 1/20 0.41
PSIP1 O75475 1/20 0.41
AXL P30530 1/20 0.41
CYP11B1 P15538 4/20 0.41
CYP17A1 P05093 2/20 0.41
CYP19A1 P11511 2/20 0.40
KIF11 P52732 1/20 0.40
DYRK1A Q13627 1/20 0.40
DYRK1B Q9Y463 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2922495 0.81 CYP2A6 (0.55) GRM5CYP2A6CYP1A2CYP3A4
SCHEMBL30694380 0.81 CYP2A6 (0.55) GRM5CYP2A6CYP1A2CYP3A4
SCHEMBL29934042 0.79 GRM5 (0.40) GRM5CYP2A6
SCHEMBL28884696 0.79 GRM5 (0.40) GRM5CYP2A6
SCHEMBL3346852 0.77 CYP11B2 (0.47) GRM5CYP11B2CYP11B1
SCHEMBL31510379 0.77 GRM5 (0.55) GRM5CYP2A6CYP1A2CYP3A4
SCHEMBL22531723 0.76 GRM5 (0.38) GRM5CYP2A6
SCHEMBL1690481 0.76 CYP11B2 (0.68) GRM5CYP2A6ALDH1A1CYP1A2CYP3A4
SCHEMBL4855910 0.75 GRM5 (0.60) GRM5CYP2A6ALDH1A1CYP1A2CYP3A4
SCHEMBL3348429 0.75 GRM5 (0.44) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed