SCHEMBL3350871

SCHEMBL3350871

O=C(NCCc1cccc(Cl)c1)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)nc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.57
TAAR1 Q96RJ0 4/20 0.48
ALDH1A1 P00352 4/20 0.48
GLA P06280 1/20 0.48
TP53 P04637 1/20 0.43
POLB P06746 1/20 0.43
MC4R P32245 2/20 0.41
TRPV1 Q8NER1 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
HIF1A Q16665 1/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40
PLAAT3 P53816 2/20 0.40
PLAAT5 Q96KN8 2/20 0.40
PLAAT2 Q9NWW9 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3348194 0.89 KCNH2 (0.63) KCNH2TAAR1POLBMC4RGAA
SCHEMBL3348171 0.88 TAAR1 (0.53) KCNH2TAAR1ALDH1A1GLATP53
SCHEMBL3346356 0.86 KCNH2 (0.57) KCNH2TAAR1ALDH1A1GLATP53
SCHEMBL3415193 0.84 KCNH2 (0.65) KCNH2TAAR1POLBMC4RPLAAT3
SCHEMBL3346386 0.82 TAAR1 (0.48) KCNH2TAAR1ALDH1A1GLATP53
SCHEMBL3353112 0.80 MC4R (0.43) KCNH2TAAR1ALDH1A1GLATP53
SCHEMBL3345900 0.80 KCNH2 (0.58) KCNH2MC4RTRPV1KDM4ELMNA
SCHEMBL3350867 0.79 KCNH2 (0.52) KCNH2TRPV1
SCHEMBL3350808 0.79 TAAR1 (0.53) TAAR1ALDH1A1GLATP53POLB
SCHEMBL3410485 0.79 MC4R (0.43) KCNH2TAAR1ALDH1A1GLATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed