SCHEMBL3352929

SCHEMBL3352929

CCCN(CCC)C(=O)CC(N)=O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
HPGD P15428 1/20 0.48
CA12 O43570 6/20 0.44
CA9 Q16790 6/20 0.44
CA2 P00918 5/20 0.44
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 1/20 0.40
APEX1 P27695 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TP53 P04637 1/20 0.38
CA1 P00915 5/20 0.37
SIGMAR1 Q99720 1/20 0.36
PKM P14618 1/20 0.35
ALOX15 P16050 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MLYCD O95822 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3621282 0.85 ALDH1A1 (0.56) ALDH1A1HPGDCA12CA9CA2
SCHEMBL5712587 0.83 CA12 (0.44) CA12CA9CA2TP53CA1
SCHEMBL10341598 0.83 CA12 (0.44) CA12CA9CA2TP53CA1
SCHEMBL11315449 0.83 CA12 (0.44) CA12CA9CA2TP53CA1
SCHEMBL2977192 0.80 LMNA (0.50) ALDH1A1CA12CA9CA2CA1
SCHEMBL16133337 0.79 ALDH1A1 (0.47) ALDH1A1HPGDCA12CA9CA2
SCHEMBL15224146 0.79 KDM5A (0.33) ALDH1A1HPGDCA12CA9CA2
SCHEMBL3351986 0.79 ALDH1A1 (0.57) ALDH1A1HPGDCA12CA9CA2
SCHEMBL7482394 0.78 ALDH1A1 (0.50) ALDH1A1HPGDCA12CA9CA2
SCHEMBL1890865 0.78 MAOA (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111071993-B Working solution solvent system 中国石油化工股份有限公司 2021-06-04 CN disclosed
CN-111071993-A Working solution solvent system 中国石油化工股份有限公司 2020-04-28 CN disclosed
CN-108026027-A substituted Malonamide compounds and their use as antibacterial agents 邱浩杰 2018-05-11 CN disclosed
US-7727997-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2010-06-01 US disclosed
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease ELAN PHARMACEUTICALS, INC. 2007-09-13 US disclosed
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US disclosed
EP-0410726-A1 S-substituted beta-thioacrylamides and their use as microbicides ROHM AND HAAS COMPANY (US) 1991-01-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease BACE1, BACE2, APP ALDH1A1 2133/4885HPGD 1390/4885CA12 4160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.