SCHEMBL3353133

SCHEMBL3353133

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1cc(Cl)cc(Cl)c1)c1cccc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.47
ROCK2 O75116 5/20 0.41
KCNQ3 O43525 2/20 0.40
KCNQ2 O43526 2/20 0.40
SLC6A4 P31645 1/20 0.39
KCNQ4 P56696 1/20 0.39
KCNQ5 Q9NR82 1/20 0.39
MTOR P42345 1/20 0.38
GPR139 Q6DWJ6 3/20 0.38
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
JAK3 P52333 1/20 0.37
CACNA1H O95180 2/20 0.37
MC4R P32245 1/20 0.37
MC5R P33032 1/20 0.37
MC3R P41968 1/20 0.37
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
PRKG1 Q13976 1/20 0.36
REN P00797 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3353036 0.92 KCNH2 (0.52) KCNH2ROCK2KCNQ3KCNQ2SLC6A4
SCHEMBL13365099 0.92 KCNH2 (0.52) KCNH2ROCK2KCNQ3KCNQ2SLC6A4
SCHEMBL13365065 0.92 KCNH2 (0.52) KCNH2ROCK2KCNQ3KCNQ2SLC6A4
SCHEMBL3353124 0.92 KCNH2 (0.52) KCNH2ROCK2KCNQ3KCNQ2SLC6A4
SCHEMBL13365101 0.88 KCNH2 (0.54) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3353138 0.88 KCNQ3 (0.52) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3353040 0.88 KCNH2 (0.48) KCNH2ROCK2KCNQ3KCNQ2SLC6A4
SCHEMBL3347954 0.86 POLB (0.54) KCNH2ROCK2POLBMAPK1PRKG1
SCHEMBL3346492 0.86 ROCK2 (0.46) KCNH2ROCK2KCNQ3KCNQ2SLC6A4
SCHEMBL3353108 0.85 KCNH2 (0.46) KCNH2ROCK2KCNQ3KCNQ2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed