SCHEMBL3346492

SCHEMBL3346492

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(Cl)cc1Cl)c1cccc(F)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.46
KCNH2 Q12809 1/20 0.43
SLC6A4 P31645 2/20 0.42
DPP4 P27487 2/20 0.41
MC4R P32245 4/20 0.39
PRCP P42785 2/20 0.37
MTOR P42345 1/20 0.37
BRS3 P32247 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
PTGER4 P35408 1/20 0.36
PTGER2 P43116 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.36
GPR139 Q6DWJ6 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3349846 0.90 ROCK2 (0.48) ROCK2KCNH2BRS3GAAHPGD
SCHEMBL13365099 0.88 KCNH2 (0.52) ROCK2KCNH2SLC6A4MC4RPRCP
SCHEMBL3353124 0.88 KCNH2 (0.52) ROCK2KCNH2SLC6A4MC4RPRCP
SCHEMBL3353036 0.88 KCNH2 (0.52) ROCK2KCNH2SLC6A4MC4RPRCP
SCHEMBL13365065 0.88 KCNH2 (0.52) ROCK2KCNH2SLC6A4MC4RPRCP
SCHEMBL3353133 0.86 KCNH2 (0.47) ROCK2KCNH2SLC6A4MC4RMTOR
SCHEMBL3353040 0.84 KCNH2 (0.48) ROCK2KCNH2SLC6A4MTORSMN1; SMN2
SCHEMBL3380842 0.83 KCNH2 (0.40) ROCK2KCNH2SLC6A4SMN1; SMN2PTGER4
SCHEMBL3353108 0.80 KCNH2 (0.46) ROCK2KCNH2KCNQ3KCNQ2
SCHEMBL13365133 0.79 ROCK2 (0.48) ROCK2SLC6A4DPP4KCNQ3KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed