SCHEMBL3358352

SCHEMBL3358352

Cc1ccc(-c2no[c]c2C(N)=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.41
GAA P10253 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KDR P35968 2/20 0.38
PDGFRB P09619 1/20 0.38
MAPK1 P28482 1/20 0.38
MAP2K4 P45985 1/20 0.38
MAPKAPK2 P49137 1/20 0.38
MAPKAPK3 Q16644 1/20 0.38
MAPK6 Q16659 1/20 0.38
MAPKAPK5 Q8IW41 1/20 0.38
KIF11 P52732 1/20 0.38
F9 P00740 1/20 0.36
KDM4E B2RXH2 3/20 0.36
MAPT P10636 2/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2795904 0.84 LMNA (0.40) IKBKBCA12CA1CA2CA9
SCHEMBL2464885 0.71
SCHEMBL105146 0.68 IKBKB (0.48) IKBKBGAAMEN1KMT2AKDR
SCHEMBL3823644 0.66 IKBKB (0.49) IKBKBGAAMEN1KMT2AKDR
SCHEMBL5981249 0.63 CA1 (0.55) MAPK1MAP2K4MAPKAPK2MAPKAPK3MAPK6
SCHEMBL20705487 0.63 CA1 (0.55) MAPK1MAP2K4MAPKAPK2MAPKAPK3MAPK6
P-Xylene SCHEMBL28147896 0.62 ALDH1A1 (0.58) GAAMEN1KMT2AKIF11NPSR1
SCHEMBL3987365 0.62 MAPT (0.49) MEN1KMT2AKDM4EMAPTRAB9A
SCHEMBL3310365 0.62 SCN9A (0.51) IKBKBGAAMEN1KMT2AKDR
SCHEMBL3081965 0.62 MKNK1 (0.40) IKBKBMEN1KMT2AKDRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9370506-B2 Modulators of aldehyde dehydrogenase and methods of use thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2016-06-21 US disclosed
US-20150182506-A1 Modulators of Aldehyde Dehydrogenase and Methods of Use Thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2015-07-02 US disclosed
US-20140343045-A1 Modulators of Aldehyde Dehydrogenase and Methods of Use Thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2014-11-20 US disclosed
US-8772295-B2 Modulators of aldehyde dehydrogenase and methods of use thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2014-07-08 US disclosed
US-20130267501-A1 Modulators of Aldehyde Dehydrogenase and Methods of Use Thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2013-10-10 US disclosed
US-8389522-B2 Modulators of aldehyde dehydrogenase and methods of use thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2013-03-05 US disclosed
WO-2010062308-A1 MODULATORS OF ALDEHYDE DEHYDROGENASE AND METHODS OF USE THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2010-06-03 WO disclosed
US-20100113423-A1 Modulators of Aldehyde Dehydrogenase and Methods of Use Thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140343045-A1 Modulators of Aldehyde Dehydrogenase and Methods of Use Thereof ALDH2, ALDH3A1, ALDH1A1 IKBKB 1378/4885GAA 63/4885MEN1 4664/4885
US-20150182506-A1 Modulators of Aldehyde Dehydrogenase and Methods of Use Thereof ALDH2, ALDH3A1, ALDH1A1 IKBKB 1378/4885GAA 63/4885MEN1 4664/4885
US-20130267501-A1 Modulators of Aldehyde Dehydrogenase and Methods of Use Thereof ALDH2, ALDH3A1, ALDH1A1 IKBKB 1378/4885GAA 63/4885MEN1 4664/4885
US-20100113423-A1 Modulators of Aldehyde Dehydrogenase and Methods of Use Thereof ALDH2, ALDH3A1, ALDH1A1 IKBKB 1378/4885GAA 63/4885MEN1 4664/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.