SCHEMBL3358739

SCHEMBL3358739

c1csc(-c2ccnc3c2ccc2c(-c4cccs4)ccnc23)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.59
GLO1 Q04760 1/20 0.50
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
TGFBR1 P36897 1/20 0.42
MAPK14 Q16539 1/20 0.42
GAA P10253 2/20 0.42
GFER P55789 1/20 0.42
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
CDK5 Q00535 2/20 0.40
CDK5R1 Q15078 2/20 0.40
CYP2E1 P05181 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2A6 P11509 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2B6 P20813 1/20 0.40
CCNB2 O95067 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28083058 0.86 TOP2A (0.49) TOP2AGLO1KDM4EALDH1A1TGFBR1
SCHEMBL28203392 0.85 TOP2A (0.48) TOP2AGLO1KDM4EALDH1A1PDE3B
SCHEMBL8087934 0.78 TGFBR1 (0.65) TOP2AKDM4EALDH1A1TGFBR1MAPK14
SCHEMBL2237236 0.78 GLO1 (0.47) TOP2AGLO1KDM4EALDH1A1GAA
SCHEMBL22523304 0.77 TOP2A (1.00) TOP2AGLO1KDM4EALDH1A1CDK2
SCHEMBL17599154 0.77 TGFBR1 (0.63) TOP2AKDM4EALDH1A1TGFBR1MAPK14
SCHEMBL28915652 0.76 GLO1 (0.56) TOP2AGLO1KDM4EALDH1A1GAA
SCHEMBL858198 0.74 AURKB (0.57) CDK2CDK5CDK5R1CCNB2CDK1
SCHEMBL29946359 0.74 AURKB (0.57) CDK2CDK5CDK5R1CCNB2CDK1
SCHEMBL498344 0.73 GLO1 (0.47) GLO1KDM4EALDH1A1GAAGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2161272-A1 Phenanthrolines BASF SE (DE) 2010-03-10 EP disclosed