SCHEMBL335918

SCHEMBL335918

COc1ccc2[nH]c(C(=O)NC(c3ccccc3)C(O)C(=O)Nc3ccc4c(N)nccc4c3)cc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F9 P00740 2/20 0.45
PYGL P06737 1/20 0.44
KDM4E B2RXH2 7/20 0.43
NPC1 O15118 5/20 0.43
RAB9A P51151 5/20 0.43
ALDH1A1 P00352 4/20 0.43
PRNP P04156 1/20 0.43
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
BCAT1 P54687 1/20 0.43
MAPT P10636 5/20 0.43
KMT2A Q03164 2/20 0.42
PLCG2 P16885 1/20 0.42
F7 P08709 2/20 0.41
F3 P13726 2/20 0.41
APP P05067 1/20 0.41
ACHE P22303 1/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL335762 0.94 PYGL (0.44) PYGLKDM4ENPC1RAB9AALDH1A1
SCHEMBL335793 0.85 F9 (0.50) F9KDM4ENPC1RAB9AALDH1A1
SCHEMBL336071 0.84 PYGL (0.45) PYGLKDM4ENPC1RAB9AALDH1A1
SCHEMBL15282234 0.82 ITK (0.38) F9KDM4EKMT2AF7F3
SCHEMBL336483 0.80 F9 (0.54) F9F7F3
SCHEMBL334902 0.79 F9 (0.49) F9NPC1ALDH1A1L3MBTL1MAPT
SCHEMBL335308 0.78 MEN1 (0.44) NPC1RAB9AL3MBTL1KMT2AMEN1
SCHEMBL335786 0.77 F9 (0.51) F9F7F3
SCHEMBL335322 0.76 F9 (0.64) F9RAB9AF7F3
SCHEMBL335183 0.76 ALDH1A1 (0.55) F9NPC1RAB9AALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097758-B2 Isoserine derivatives for use as coagulation factor IXa inhibitors SANOFI-AVENTIS (FR) 2012-01-17 US claimed