SCHEMBL3362291

SCHEMBL3362291

C[C@]12CCC(O)CC1CC(=O)[C@@H]1[C@@H]2CC[C@]2(C)C(=O)CC[C@@H]12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 1.00
RIN1 Q13671 1/20 1.00
GPBAR1 Q8TDU6 5/20 0.65
LMNA P02545 4/20 0.65
CYP3A4 P08684 4/20 0.65
MEN1 O00255 4/20 0.65
KMT2A Q03164 4/20 0.65
SHBG P04278 3/20 0.65
SERPINA6 P08185 3/20 0.65
PMP22 Q01453 2/20 0.65
G6PD P11413 2/20 0.65
TSHR P16473 2/20 0.65
AKR1B10 O60218 2/20 0.65
AKR1B1 P15121 2/20 0.65
MAPK1 P28482 1/20 0.65
HSD17B3 P37058 1/20 0.65
CYP2D6 P10635 1/20 0.65
NFKB1 P19838 1/20 0.65
CYP2C19 P33261 1/20 0.65
SLC10A2 Q12908 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7062423 1.00 ABL1 (1.00) ABL1RIN1GPBAR1LMNACYP3A4
SCHEMBL4339194 1.00 ABL1 (1.00) ABL1RIN1GPBAR1LMNACYP3A4
SCHEMBL2509859 1.00 ABL1 (1.00) ABL1RIN1GPBAR1LMNACYP3A4
SCHEMBL12057060 1.00 ABL1 (1.00) ABL1RIN1GPBAR1LMNACYP3A4
SCHEMBL2509858 1.00 ABL1 (1.00) ABL1RIN1GPBAR1LMNACYP3A4
SCHEMBL5445469 0.83 ABL1 (0.70) ABL1RIN1GPBAR1LMNACYP3A4
SCHEMBL1115615 0.83 ABL1 (0.70) ABL1RIN1GPBAR1LMNACYP3A4
SCHEMBL6881931 0.83 ABL1 (0.70) ABL1RIN1GPBAR1LMNACYP3A4
SCHEMBL6448971 0.83 ABL1 (0.70) ABL1RIN1GPBAR1LMNACYP3A4
SCHEMBL6876271 0.83 ABL1 (0.70) ABL1RIN1GPBAR1LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100009970-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF VIRAL DISEASES COMBINATORX (SINGAPORE) PTE. LTD. (SG) 2010-01-14 US disclosed
EP-2004669-A1 AZAHETEROCYCLYL DERIVATIVES OF ANDROSTANES AND ANDROSTENES AS MEDICAMENTS FOR CARDIOVASCULAR DISORDERS SIGMA-TAU Industrie Farmaceutiche Riunite S.p.A. (IT) 2008-12-24 EP disclosed
EP-2004668-A2 AMINO DERIVATIVES OF ANDROSTANES AND ANDROSTENES AS MEDICAMENTS FOR CARDIOVASCULAR DISORDERS SIGMA-TAU Industrie Farmaceutiche Riunite S.p.A. (IT) 2008-12-24 EP disclosed
US-20080161324-A1 Compositions and methods for treatment of viral diseases EXCRX (SINGAPORE) PTE. LTD. (F.K.A. COMBINATORX (SINGAPORE) PTE LTD.) (SG) 2008-07-03 US disclosed
WO-2008033466-A2 COMPOSITIONS AND METHODS FOR TREATMENT OF VIRAL DISEASES COMBINATORX (SINGAPORE) PRE. LTD. (SG) 2008-03-20 WO disclosed
WO-2007118830-A1 AZAHETEROCYCLYL DERIVATIVES OF ANDROSTANES AND ANDROSTENES AS MEDICAMENTS FOR CARDIOVASCULAR DISORDERS SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2007-10-25 WO disclosed
WO-2007118832-A2 AMINO DERIVATIVES OF ANDROSTANES AND ANDROSTENES AS MEDICAMENTS FOR CARDIOVASCULAR DISORDERS SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2007-10-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100009970-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF VIRAL DISEASES HTR1A, HTR3B, HTR3A ABL1 992/4885RIN1 4338/4885GPBAR1 589/4885
US-20080161324-A1 Compositions and methods for treatment of viral diseases HAVCR2, EIF2AK2, RNASE1 ABL1 310/4885RIN1 4331/4885GPBAR1 470/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.