SCHEMBL3363185

SCHEMBL3363185

COc1cc2c(CC(=O)NC(C)c3cccnc3)cnc(CNC(=O)OC(C)(C)C)c2cc1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.39
CYP3A4 P08684 5/20 0.38
DPP4 P27487 2/20 0.37
KMT2A Q03164 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
MEN1 O00255 1/20 0.37
CYP2C19 P33261 1/20 0.37
ADORA2B P29275 1/20 0.37
ROCK2 O75116 1/20 0.37
PRKG1 Q13976 1/20 0.37
TSHR P16473 2/20 0.36
ABCB1 P08183 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
RECQL P46063 1/20 0.36
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362959 0.80 DPP4 (0.40) DPP4
SCHEMBL3363192 0.79 CYP3A4 (0.41) NAMPTCYP3A4DPP4KMT2ANPSR1
SCHEMBL3361880 0.79 DPP4 (0.47) DPP4
SCHEMBL3361314 0.78 NPC1 (0.44) DPP4ALDH1A1TP53MAPTHSD17B10
SCHEMBL3362189 0.77 DPP4 (0.43) DPP4L3MBTL1TP53
SCHEMBL5746285 0.74 GFPT1 (0.48) ABCB1L3MBTL1HSD17B10
SCHEMBL3361800 0.73 CTSL (0.43) DPP4KMT2AMEN1L3MBTL1TP53
SCHEMBL3362196 0.73 DPP4 (0.46) DPP4
SCHEMBL6110619 0.72 GFPT1 (0.41) L3MBTL1HSD17B10
SCHEMBL3360434 0.72 DPP4 (0.41) DPP4KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed