SCHEMBL3366103

SCHEMBL3366103

CCN(Cc1ccccc1)C(=O)Nc1cnc(CNC(=O)OC(C)(C)C)c2c(OC)cc(OC)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.40
HTT P42858 2/20 0.40
GAA P10253 1/20 0.40
TRPV1 Q8NER1 1/20 0.39
ROCK2 O75116 5/20 0.38
PTPN1 P18031 1/20 0.36
DPP4 P27487 2/20 0.35
ALOX15 P16050 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
ROCK1 Q13464 1/20 0.34
CDC42BPA Q5VT25 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7723483 0.93 GAA (0.40) TSHRHTTGAAROCK2DPP4
SCHEMBL7716634 0.91 ABCC1 (0.38) TSHRHTTGAAROCK2PTPN1
SCHEMBL3362425 0.85 DPP4 (0.50) TSHRHTTGAATRPV1ROCK2
SCHEMBL3362011 0.85 DPP4 (0.40) TSHRDPP4NPSR1CTSLKMT2A
SCHEMBL3361514 0.84 GAA (0.44) TSHRHTTGAATRPV1ROCK2
SCHEMBL3361319 0.83 GAA (0.44) HTTGAASMN1; SMN2MEN1KMT2A
SCHEMBL3361777 0.82 TP53 (0.41) TSHRROCK2DPP4ROCK1MEN1
SCHEMBL3365615 0.81 DPP4 (0.41) HTTGAAROCK2PTPN1DPP4
SCHEMBL3360962 0.79 DPP4 (0.41) GAADPP4KMT2A
SCHEMBL3361886 0.78 DPP4 (0.41) TSHRHTTDPP4ALOX15SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed