SCHEMBL3362011

SCHEMBL3362011

COc1cc(OC)c2c(CNC(=O)OC(C)(C)C)ncc(NC(=O)N(C)C)c2c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.40
ABCB1 P08183 2/20 0.37
GFER P55789 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DYRK1A Q13627 2/20 0.35
MAPKAPK2 P49137 3/20 0.33
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32
SKP2 Q13309 1/20 0.32
CTSL P07711 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
KMT2A Q03164 1/20 0.32
PDPK1 O15530 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7716634 0.88 ABCC1 (0.38) DPP4CKS1BSKP1SKP2CTSL
SCHEMBL3360962 0.88 DPP4 (0.41) DPP4ABCB1GFERHSD17B10L3MBTL1
SCHEMBL3361319 0.85 GAA (0.44) HSD17B10L3MBTL1ALDH1A1KMT2A
SCHEMBL3366103 0.85 TSHR (0.40) DPP4CTSLTSHRNPSR1KMT2A
SCHEMBL7723483 0.84 GAA (0.40) DPP4ABCB1DYRK1AALDH1A1TSHR
SCHEMBL3362437 0.83 DPP4 (0.45) DPP4ABCB1GFERHSD17B10L3MBTL1
SCHEMBL3363099 0.82 DPP4 (0.49) DPP4ABCB1GFERHSD17B10L3MBTL1
SCHEMBL3363078 0.81 DPP4 (0.58) DPP4ALDH1A1
SCHEMBL3362364 0.79 ABCB1 (0.40) DPP4ABCB1HSD17B10DYRK1AALDH1A1
SCHEMBL3360966 0.79 DPP4 (0.41) DPP4ABCB1GFERHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed