SCHEMBL3366423

SCHEMBL3366423

Cc1cc(C#N)cc(C)c1-c1ccnc(N)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.43
NOS1 P29475 3/20 0.43
NOS2 P35228 3/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
DYRK1A Q13627 4/20 0.41
GSK3B P49841 1/20 0.40
EGLN2 Q96KS0 4/20 0.40
MET P08581 1/20 0.39
AAK1 Q2M2I8 2/20 0.39
CDC7 O00311 1/20 0.39
CDK2 P24941 1/20 0.39
S1PR1 P21453 1/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
GRM5 P41594 1/20 0.36
KCNH2 Q12809 1/20 0.36
ROCK1 Q13464 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3366217 0.81 KCNH2 (0.52) NOS3NOS1NOS2KDM4EMEN1
SCHEMBL3361839 0.81 GRM5 (0.43) EGLN2CDK2GRM5
SCHEMBL3366055 0.79 NOS3 (0.52) NOS3NOS1NOS2KDM4EMEN1
SCHEMBL3397985 0.76 DYRK1A (0.54) DYRK1AGSK3BEGLN2AAK1CDC7
SCHEMBL29432635 0.76 DYRK1A (0.54) DYRK1AGSK3BEGLN2AAK1CDC7
SCHEMBL23809618 0.73 DYRK1A (0.45) NOS3NOS1NOS2KDM4EMEN1
SCHEMBL18998664 0.73 CLK4 (0.59) DYRK1AGSK3BCDC7CDK2GRM5
SCHEMBL312451 0.73
SCHEMBL31294130 0.73
SCHEMBL3360845 0.72 EGLN2 (0.48) DYRK1AGSK3BEGLN2METAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed