SCHEMBL3367593

SCHEMBL3367593

CNC(=O)Oc1c2cccc(-c3ccc(Cl)cc3Cl)c2nn1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 11/20 0.44
CHRM3 P20309 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
GAA P10253 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
NFKB1 P19838 1/20 0.36
STAT3 P40763 1/20 0.36
STAT1 P42224 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CNR1 P21554 2/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364228 0.88 CRHR1 (0.46) CRHR1KDM4EALDH1A1HPGDGAA
SCHEMBL3363623 0.87 CRHR1 (0.42) CRHR1CNR1DPP4DPP8
SCHEMBL3367997 0.85 CRHR1 (0.44) CRHR1KDM4EALDH1A1GAANPC1
SCHEMBL3368609 0.83 KDM4E (0.45) CRHR1KDM4ELMNASMN1; SMN2CNR1
SCHEMBL3366121 0.81 CRHR1 (0.48) CRHR1
SCHEMBL3364408 0.81 CRHR1 (0.46) CRHR1ALDH1A1HPGDLMNARAB9A
SCHEMBL3362477 0.80 CRHR1 (0.47) CRHR1KDM4E
SCHEMBL3366050 0.79 CRHR1 (0.46) CRHR1CHRM3KDM4EALDH1A1HPGD
SCHEMBL3367673 0.79 S1PR4 (0.38) CRHR1KDM4EALDH1A1HPGDGAA
SCHEMBL3364735 0.79 CRHR1 (0.51) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed