SCHEMBL3367918

SCHEMBL3367918

O=C(O)C1CN=C(c2ccc(Br)cc2O)S1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.35
PKM P14618 1/20 0.35
BCL2 P10415 1/20 0.35
MCL1 Q07820 1/20 0.35
SRD5A1 P18405 1/20 0.34
SRD5A2 P31213 1/20 0.34
EDNRB P24530 2/20 0.33
EDNRA P25101 2/20 0.33
ALOX15 P16050 2/20 0.33
CES2 O00748 1/20 0.33
GALR3 O60755 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CASP1 P29466 1/20 0.33
CYP2C19 P33261 1/20 0.33
CSNK2A1 P68400 1/20 0.32
GRK6 P43250 1/20 0.32
IDO1 P14902 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3368482 0.91 HPGD (0.40) HPGDPKMBCL2MCL1EDNRB
SCHEMBL3369371 0.85 TYR (0.37) HPGDCES2CSNK2A1MAOBMAPT
SCHEMBL3370061 0.84 PKM (0.33) HPGDPKMBCL2MCL1MAOA
SCHEMBL3372129 0.82 HTR2B (0.46) HPGDPKMHTR2BTP53MAPT
SCHEMBL10066500 0.70
SCHEMBL2114802 0.66 HCAR2 (0.35) PKMMAPTATM
SCHEMBL2114806 0.66 HCAR2 (0.35) PKMMAPTATM
SCHEMBL31396259 0.65 EDNRB (0.41) HPGDPKMBCL2MCL1SRD5A1
SCHEMBL2115910 0.64 KMO (0.44) CYP1A2CYP2C9CYP2C19KDM4EGAA
SCHEMBL29502821 0.63 ALOX15 (0.57) HPGDBCL2MCL1ALOX15CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010018458-A2 PHENOL DERIVATIVES AND METHODS OF USE THEREOF CRYSTALGENOMICS, INC. (KR) 2010-02-18 WO claimed
WO-2010018458-A2 PHENOL DERIVATIVES AND METHODS OF USE THEREOF CRYSTALGENOMICS, INC. (KR) 2010-02-18 WO disclosed