SCHEMBL3373184

SCHEMBL3373184

O=C(O)C(=Cc1ccccc1)c1cncnc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 4/20 0.67
AKR1C3 P42330 4/20 0.51
AKR1C2 P52895 3/20 0.49
KMT2A Q03164 5/20 0.47
MEN1 O00255 4/20 0.47
POLB P06746 2/20 0.47
PTGS2 P35354 1/20 0.47
ALDH1A1 P00352 4/20 0.45
HCAR2 Q8TDS4 1/20 0.45
MAPT P10636 3/20 0.45
KDM4E B2RXH2 2/20 0.45
HPGD P15428 2/20 0.45
HTT P42858 2/20 0.45
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3373182 1.00 AKR1C1 (0.67) AKR1C1AKR1C3AKR1C2KMT2AMEN1
SCHEMBL19031900 0.87 CYP11B2 (0.53) AKR1C1KMT2AMEN1ALDH1A1HCAR2
SCHEMBL19031899 0.87 CYP11B2 (0.53) AKR1C1KMT2AMEN1ALDH1A1HCAR2
SCHEMBL3373196 0.86 AKR1C1 (0.67) AKR1C1AKR1C3AKR1C2KMT2AMEN1
SCHEMBL8646375 0.83 AKR1C1 (0.68) AKR1C1AKR1C3AKR1C2KMT2AMEN1
SCHEMBL8646379 0.83 AKR1C1 (0.68) AKR1C1AKR1C3AKR1C2KMT2AMEN1
SCHEMBL39275 0.81 AKR1C1 (1.00) AKR1C1AKR1C3AKR1C2KMT2AMEN1
SCHEMBL181529 0.81 AKR1C1 (1.00) AKR1C1AKR1C3AKR1C2KMT2AMEN1
SCHEMBL290469 0.81 AKR1C1 (1.00) AKR1C1AKR1C3AKR1C2KMT2AMEN1
SCHEMBL19031901 0.80 ALDH1A1 (0.51) AKR1C1KMT2AMEN1ALDH1A1HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed