SCHEMBL3373190

SCHEMBL3373190

O=C(O)C=C(c1ccccc1)c1cncnc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.47
HCAR2 Q8TDS4 2/20 0.47
TBXAS1 P24557 15/20 0.43
ALDH1A1 P00352 1/20 0.41
APP P05067 1/20 0.41
GAA P10253 1/20 0.41
HCAR3 P49019 1/20 0.41
TBXA2R P21731 4/20 0.40
PLOD2 O00469 1/20 0.40
CYP19A1 P11511 1/20 0.40
CYP11B2 P19099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28141157 0.90 BCAT2 (0.43) BCAT2TBXAS1ALDH1A1GAAPLOD2
SCHEMBL63954 0.84 CES1 (0.50) ALDH1A1
Hydrochloric Acid SCHEMBL6166969 0.82 TBXAS1 (0.59) HCAR2TBXAS1ALDH1A1APPGAA
Hydrochloric Acid SCHEMBL6166975 0.82 TBXAS1 (0.59) HCAR2TBXAS1ALDH1A1APPGAA
Hydrochloric Acid SCHEMBL6167657 0.82 TBXAS1 (0.59) HCAR2TBXAS1ALDH1A1APPGAA
Hydrochloric Acid SCHEMBL4398755 0.82 NFE2L2 (0.48) ALDH1A1
SCHEMBL8937507 0.81 KMT2A (0.61) TBXAS1ALDH1A1PLOD2CYP19A1CYP11B2
SCHEMBL8937512 0.81 KMT2A (0.61) TBXAS1ALDH1A1PLOD2CYP19A1CYP11B2
SCHEMBL8937855 0.81 KMT2A (0.61) TBXAS1ALDH1A1PLOD2CYP19A1CYP11B2
SCHEMBL16464023 0.75 HCAR2 (0.53) HCAR2TBXAS1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed