SCHEMBL3373560

SCHEMBL3373560

CCCCC(=O)NC1(C(=O)NCc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)CCCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 2/20 0.46
CTSB P07858 2/20 0.43
CTSS P25774 2/20 0.43
BDKRB1 P46663 2/20 0.40
AGTR1 P30556 3/20 0.39
AGTR2 P50052 3/20 0.39
CTSL P07711 2/20 0.38
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
POLB P06746 2/20 0.36
ABCC3 O15438 1/20 0.36
ABCC4 O15439 1/20 0.36
ABCB11 O95342 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
EDNRA P25101 1/20 0.36
MAPK1 P28482 1/20 0.36
HTR2B P41595 1/20 0.36
PDE3A Q14432 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4609709 0.86 LTB4R2 (0.60) LTB4R2BDKRB1CYP3A4CYP2C19POLB
SCHEMBL10027906 0.80 LTB4R2 (0.58) LTB4R2CTSBCTSSBDKRB1AGTR1
SCHEMBL14038695 0.80 LTB4R2 (0.38) LTB4R2AGTR1AGTR2CYP3A4ABCC3
SCHEMBL3169268 0.79 CTSB (0.49) LTB4R2CTSBCTSSBDKRB1AGTR1
SCHEMBL2959 0.79 AGTR1 (0.47) LTB4R2AGTR1AGTR2ABCB11
SCHEMBL3370402 0.78 AGTR1 (0.46) LTB4R2CTSBCTSSBDKRB1AGTR1
SCHEMBL9672280 0.78 CTSB (0.51) LTB4R2CTSBCTSSBDKRB1AGTR1
SCHEMBL8472336 0.77 AGTR1 (0.37) LTB4R2AGTR1AGTR2CYP3A4ABCC3
SCHEMBL5592312 0.76 LTB4R2 (0.45) LTB4R2AGTR1ABCB11
SCHEMBL5489422 0.76 LTB4R2 (0.42) LTB4R2AGTR1AGTR2HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113933414-B Method for detecting organic impurities in amlodipine besylate composite preparation 株洲千金药业股份有限公司 2023-07-07 CN claimed
CN-111053910-A Composition comprising fatty acid or derivative thereof and disubstituted biphenyl derivative 黄泳华 2020-04-24 CN claimed
CN-118243800-A Method for measuring related substances of irbesartan amlodipine tablets 珠海润都制药股份有限公司 2024-06-25 CN disclosed
CN-111053910-A Composition comprising fatty acid or derivative thereof and disubstituted biphenyl derivative 黄泳华 2020-04-24 CN disclosed
EP-2194050-A1 A new process for the preparation of irbesartan KRKA, tovarna zdravil, d.d., Novo mesto (SI) 2010-06-09 EP disclosed