SCHEMBL3370402

SCHEMBL3370402

CCCCC(=O)NC1(C(=O)NCc2ccc(-c3ccccc3-c3nnnn3C(c3ccccc3)(c3ccccc3)c3ccccc3)cc2)CCCC1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 4/20 0.46
AGTR2 P50052 2/20 0.46
LTB4R2 Q9NPC1 2/20 0.44
AGT P01019 2/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
ACHE P22303 1/20 0.38
BDKRB1 P46663 2/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
POLB P06746 2/20 0.35
HPGD P15428 1/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3948155 0.87 LTB4R2 (0.57) AGTR1AGTR2LTB4R2AGTPOLB
SCHEMBL13679199 0.80 AGTR1 (0.47) AGTR1AGTR2LTB4R2AGTACHE
SCHEMBL3373560 0.78 LTB4R2 (0.46) AGTR1AGTR2LTB4R2CTSBCTSS
SCHEMBL4735569 0.76 SOAT1 (0.47) AGTR1AGTR2POLBHPGD
SCHEMBL10027906 0.76 LTB4R2 (0.58) AGTR1AGTR2LTB4R2CTSBCTSS
SCHEMBL9541811 0.75 AGTR1 (0.50) AGTR1AGTR2AGT
SCHEMBL3169268 0.75 CTSB (0.49) AGTR1AGTR2LTB4R2CTSBCTSS
SCHEMBL9084585 0.75 AGTR1 (0.47) AGTR1AGTR2LTB4R2AGT
SCHEMBL489527 0.75 AGTR1 (0.49) AGTR1AGTR2AGTCYP2C19
SCHEMBL9413763 0.74 AGTR1 (0.45) AGTR1AGTR2AGT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2194050-A1 A new process for the preparation of irbesartan KRKA, tovarna zdravil, d.d., Novo mesto (SI) 2010-06-09 EP disclosed