SCHEMBL3374189

SCHEMBL3374189

COc1ccc(C2=CC(=O)N=N2)cc1OC1Cc2ccccc2C1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 12/20 0.58
PDE4A P27815 10/20 0.58
PDE4C Q08493 10/20 0.58
PDE4D Q08499 10/20 0.58
NPY5R Q15761 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3375194 0.84 PDE4A (0.56) PDE4BPDE4APDE4CPDE4D
SCHEMBL3373175 0.79 PDE4D (0.50) PDE4BPDE4APDE4CPDE4D
SCHEMBL3373535 0.79 PDE4A (0.50) PDE4BPDE4APDE4CPDE4D
SCHEMBL3374398 0.78 PDE4B (0.57) PDE4BPDE4APDE4CPDE4D
SCHEMBL3375187 0.76 PDE4B (0.57) PDE4BPDE4APDE4CPDE4D
SCHEMBL3374185 0.75 KDM4E (0.64) PDE4BPDE4APDE4CPDE4DNPY5R
SCHEMBL7361110 0.74 PDE4B (0.56) PDE4BPDE4APDE4CPDE4DNPY5R
SCHEMBL497890 0.74 PDE4B (0.57) PDE4BPDE4APDE4CPDE4DNPY5R
SCHEMBL7355624 0.74 PDE4B (0.57) PDE4BPDE4APDE4CPDE4DNPY5R
SCHEMBL3374953 0.73 PDE4B (0.48) PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100324091-A1 Pyrazolone Derivative KOWA COMPANY, LTD. (JP) 2010-12-23 US disclosed
EP-2172458-A1 PYRAZOLONE DERIVATIVE Kowa Company, Ltd. (JP) 2010-04-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100324091-A1 Pyrazolone Derivative SERPINE1, SERPINC1, TFPI PDE4B 1700/4885PDE4A 1796/4885PDE4C 2308/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.